Receptor Membrane Products for Screening
Caliper offers GPCR, ion channel, nuclear receptor, and other receptor membrane reagents for screening. All receptor membranes are derived from either human recombinant or human cell lines expressing the receptor.
Our ready-to-use preparations come with its pharmacological evaluation including KD/Bmax values and graphical representations of reference curve(s) with Ki values for each lot number. Assay specification sheets outlining basic assay parameters and conditions are also included with each shipment. In addition, these same membrane preparations are used at Caliper’s Discovery Alliances & Services division, in vitro assay services, to ensure continued QA/QC validation and the highest quality materials.
Custom receptor preparations are available upon request.
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Receptor Membrane Products
- Adenosine Transporter Receptor Membranes
- Adrenergic, Alpha 2A Receptor Membranes
- Adrenergic, Alpha 2B Receptor Membranes
- Adrenergic, Beta 1 Receptor Membranes
- Adrenergic, Beta 2 Receptor Membranes
- Adrenergic, Beta 3 Receptor Membranes
- Anaphylatoxin, Complement C5a Receptor Membranes
- Androgen (Testosterone) Receptor Membranes
- Angiotensin II, Type I Receptor Membranes
- Benzodiazepine, peripheral Receptor Membranes
- CHO-K1 Control Receptor Membranes
- Dopamine, D1 Receptor Membranes
- Endothelin, ETA Receptor Membranes
- Estrogen Receptor Membranes
- HEK 293 Control Receptor Membranes
- Neuropeptide, NPY2 Receptor Membranes
- Nicotinic, aBnTx insensitive Receptor Membranes
- Progesterone
- Serotonin Transporter Receptor Membranes
- Serotonin, 5HT3 Receptor Membranes

